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List of Adenosine Receptor Regulating Nucleoside Analogues

Adenosine A1 agonists

Structure Activity


EC50 (hA1R) up to 0.1 nM

Ki up to 28 nM

B. Preti, A. Suchankova, G. Deganutti, M. Leuenberger, K. Barkan, I. Manulak, X. Huang, S. Carvalho, G. Ladds, M. Lochner Discovery and Structure–Activity Relationship Studies of Novel Adenosine A1 Receptor-Selective Agonists J. Med. Chem. 2022 10.1021/acs.jmedchem.2c01414